BI-9321 (trihydrochloride)
Catalogue number:
HY-114208A-25mg
Supplier:
Size:
25 mg _$$_
Product is available in:
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:
2387510-87-2
Purity:
98.4
Molecular Formula:
C22H24Cl3FN4
Molecular Weight:
469.81
- Data sheet: View or download
- MSDS: View or download
- Protocol: View or download
Product Description:
BI-9321 trihydrochloride is a potent, selective and cellular active nuclear receptor-binding SET domain 3 (NSD3)-PWWP1 domain antagonist with a Kd value of 166 nM. BI-9321 trihydrochloride is inactive against NSD2-PWWP1 and NSD3-PWWP2. BI-9321 trihydrochloride specifically disrupts histone interactions of the NSD3-PWWP1 domain with an IC50 of 1.2 µM in U2OS cells[1].
Storage Temperature:
4°C (Powder, stored under nitrogen, away from moisture)