This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:
1643462-64-9
Purity:
99.87
Molecular Weight:
391.34
Alternative Names:
(Rac)-PF-06649751; (Rac)-CVL-751
- Data sheet: View or download
- MSDS: View or download
- Protocol: View or download
Product Description:
(Rac)-Tavapadon ((Rac)-PF-06649751) is a potent and selective noncatechol dopamine D1 receptor agonist. (Rac)-Tavapadon displays potent full agonism in the GS activation assay as well as partial agonism in the β-arrestin2 recruitment assay (GS-cAMP, EC50=0.8 nM; β-arrestin2, EC50=68 nM). (Rac)-Tavapadon has antiparkinsonian activity[1].
Storage Temperature:
-20°C, 3 years; 4°C, 2 years (Powder)