VU0134992 (hydrochloride)
Catalogue number:
HY-122560A-1ml
Supplier:
Size:
1 ml
Product is available in:
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:
1052515-91-9
Purity:
98.34
Molecular Weight:
447.84
- Data sheet: View or download
- MSDS: View or download
- Protocol: View or download
Product Description:
VU0134992 hydrochloride is the first subtype-preferring, orally active and selective Kir4.1 potassium channel pore blocker, with an IC50 of 0.97 µM. VU0134992 hydrochloride is 9-fold selective for homomeric Kir4.1 over Kir4.1/5.1 concatemeric channels (IC50=9 µM) at -120 mV[1].
Storage Temperature:
4°C (Powder, sealed storage, away from moisture)