MS1943
Catalogue number:
HY-133129-5mg
Supplier:
Size:
5 mg
Product is available in:
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:
2225938-17-8
Purity:
98.02
Molecular Weight:
718.93
- Data sheet: View or download
- MSDS: View or download
- Protocol: View or download
Product Description:
MS1943 is a first-in-class, orally bioavailable EZH2 selective degrader, with an IC50 of 120 nM. MS1943 significantly reduces EZH2 protein levels in numerous triple-negative breast cancer (TNBC) and other cancer and noncancerous cell lines. MS1943 effectively blocks proliferation of multiple TNBC and other cancer cell lines[1].
Storage Temperature:
-20°C, 3 years; 4°C, 2 years (Powder)