(E/Z)-GSK5182
Catalogue number:
HY-111226A-1ml
Supplier:
Size:
1 ml
Product is available in:
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:
2699724-40-6
Purity:
99.17
Molecular Weight:
417.54
- Data sheet: View or download
- MSDS: View or download
- Protocol: View or download
Product Description:
(E/Z)-GSK5182 is a racemic compound of (E)-GSK5182 and (Z)-GSK5182 isomers. GSK5182 is a highly selective and orally active inverse agonist of estrogen-related receptor γ (ERRγ) with an IC50 of 79 nM[1]. GSK5182 also induces reactive oxyen species (ROS) generation in hepatocellular carcinoma[1][2][3].
Storage Temperature:
-20°C, 3 years; 4°C, 2 years (Powder)