Gartisertib
Catalogue number:
HY-136270-10mg
Supplier:
Size:
10 mg
Product is available in:
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:
1613191-99-3
Purity:
99.76
Molecular Weight:
541.55
Alternative Names:
VX-803; M4344; ATR inhibitor 2
- Data sheet: View or download
- MSDS: View or download
- Protocol: View or download
Product Description:
Gartisertib (VX-803) is an ATP-competitive, orally active, and selective ATR inhibitor, with a Ki of <150 pM. Gartisertib potently inhibits ATR-driven phosphorylated checkpoint kinase-1 (Chk1) phosphorylation with an IC50 of 8 nM. Antitumor activity[1][2].
Storage Temperature:
-20°C, 3 years; 4°C, 2 years (Powder)