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CKI-7 (free base)

Catalogue number:
HY-133028-5mg
Supplier:
Size:
5 mg _$$_
Product is available in:
  • UK
  • Ireland
  • Europe
  • USA
  • Rest of World
£107.00 Shipping is calculated in checkout
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:

120615-25-0

Purity:

99.34

Molecular Formula:

C11H12ClN3O2S

Molecular Weight:

285.75

Product Description:

CKI-7 free base is a potent and ATP-competitive casein kinase 1 (CK1) inhibitor with an IC50 of 6 µM and a Ki of 8.5 µM. CKI-7 free base is a selective Cdc7 kinase inhibitor. CKI-7 free base also inhibits SGK, ribosomal S6 kinase-1 (S6K1) and mitogen- and stress-activated protein kinase-1 (MSK1). CKI-7 free base has a much weaker effect on casein kinase II and other protein kinases[1][2][3][4].

Storage Temperature:

-20°C, 3 years; 4°C, 2 years (Powder)

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