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ML-230

Catalogue number:
CAY32552-10 mg
Supplier:
Size:
10 mg
Product is available in:
  • UK
  • Ireland
  • Europe
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  • Rest of World
£820.00 Estimated delivery Wed 7 Aug
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This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:

1776055-05-0

Purity:

≥98%

Formulation:

A crystalline solid

Molecular Weight:

439.5

Alternative Names:

3-furanyl[4-[5-(2-furanyl)-2-phenylpyrazolo[1,5-a]pyrimidin-7-yl]-1-piperazinyl]-methanone, cid-44640177

Product Description:

An inhibitor of ABCG2; selectively inhibits JC-1 efflux in Ig-MXP3 cells overexpressing ABCG2 over Jurkat cells overexpressing ABCB1 (IC50s = 0.13 and 4.65 µM, respectively); intratumoral injection with topotecan, reduces tumor size in an IGROV-1/T8 mouse xenograft model at 100 nM

Storage Temperature:

-20°C

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