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ML-133 (hydrochloride)

Catalogue number:
CAY31232-10 mg
Supplier:
Size:
10 mg
Product is available in:
  • UK
  • Ireland
  • Europe
  • USA
  • Rest of World
£227.00 Estimated delivery Tue 6 Aug
Shipping is calculated in checkout
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:

1222781-70-5

Purity:

≥98%

Formulation:

A crystalline solid

Molecular Weight:

313.8

Alternative Names:

n-[(4-methoxyphenyl)methyl]-1-naphthalenemethanamine, monohydrochloride

Product Description:

A Kir2 channel inhibitor (IC50s = 1.8, 2.8, 2,9, and 2.6 µM for Kir2.1, Kir2.2, Kir2.3, and Kir2.6, respectively); selective for Kir2 channels over Kir1.1 and Kir4.1 channels (IC50s = 33 and 76 µM, respectively); prevents the development of dynamic, but not punctate, mechanical allodynia in a mouse model of spared nerve injury at 10 and 30 nmol/animal

Storage Temperature:

-20°C

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