Adiphenine (hydrochloride)
Catalogue number:
CAY31124-10 g
Supplier:
Size:
10 g
Product is available in:
£47.00
Estimated delivery Tue 6 Aug
Shipping is calculated in checkout
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This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:
50-42-0
Purity:
≥98%
Formulation:
A crystalline solid
Molecular Weight:
347.9
Alternative Names:
α-phenyl-benzeneacetic acid, 2-(diethylamino)ethyl ester, monohydrochloride, nsc 129224, spasmolytin, trasentin
- Data sheet: View or download
- MSDS: View or download
Product Description:
An anticholinergic agent; a nAChR antagonist (IC50s = 1.8, 3.7, and 6.3 µM for the α3β4, α4β2, and α4β4 subunit-containing receptors, respectively), as well as muscarinic acetylcholine receptors (Ki = 0.44 µM); inhibits ACh-induced contractions in isolated guinea pig ileum in a concentration-dependent manner; prevents tonic hindlimb extension in a mouse model of seizures induced by MES (ED50 = 62 mg/kg); protects against organophosphate-induced lethality in mice (PD50 = 3.3 mg/kg)
Storage Temperature:
-20°C