Atipamezole
Catalogue number:
CAY34289-50 mg
Supplier:
Size:
50 mg
Product is available in:
£89.00
Estimated delivery Wed 7 Aug
Shipping is calculated in checkout
Shipping is calculated in checkout
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:
104054-27-5
Purity:
≥98%
Formulation:
A solid
Molecular Weight:
212.3
Alternative Names:
5-(2-ethyl-2,3-dihydro-1h-inden-2-yl)-1h-imidazole, mpv 1248
- Data sheet: View or download
- MSDS: View or download
Product Description:
An α2A-AR antagonist (Ki = 1.86 nM); selective for α2A-ARs over α2B- and α1-ARs (Kis = 1,949.83 and 13,300 nM, respectively), as well as over 40 receptors, ion channels, and transporters (IC50s = 540->10,000 nM); reverses medetomidine-induced bradycardia and sedation in dogs at 0.04, 0.08, and 1.2 mg/kg; enhances apomorphine- or L-DOPA-induced contralateral circling behavior and prolongs the duration of action of L-DOPA in a rat model of Parkinson’s disease at 0.3 mg/kg
Storage Temperature:
-20°C