This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:
2543545-44-2
Purity:
98.49
Molecular Weight:
449.48
- Data sheet: View or download
- MSDS: View or download
- Protocol: View or download
Product Description:
LT052 is a highly selective BET BD1 inhibitor with an IC50 of 87.7 nM. LT052 exhibits nanomolar BRD4 BD1 potency and 138-fold selectivity over BRD4 BD2 (IC50=12.130 µM). LT052 has anti-inflammatory activity and can be used for acute gout arthritis research[1].
Storage Temperature:
-20°C, 3 years; 4°C, 2 years (Powder)