TAK-683 (acetate)
Catalogue number:
HY-P2161B-1mg
Supplier:
Size:
1 mg
Product is available in:
Purity:
98.97
Molecular Weight:
1358.5
- Data sheet: View or download
- MSDS: View or download
- Protocol: View or download
Product Description:
TAK-683 acetate is a potent full KISS1 receptor (KISS1R) agonist (IC50=170 pM) with improved metabolic stability. TAK-683 acetate is a nonapeptide metastin analog, exhibits agonistic activities to KISS1R with EC50 values of 0.96 nM and 1.6 nM for human and rat, respectively[1]. TAK-683 acetate depletes GnRH in the hypothalamus and reduces plasma FSH, LH, and testosterone levels in vivo, it has the potential for the study of hormone-dependent prostate cancer[1][2][4].
Storage Temperature:
-80°C, 2 years; -20°C, 1 year (Powder, sealed storage, away from moisture and light, under nitrogen)