This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:
357425-68-4
Purity:
99.74
Molecular Formula:
C12H12F3N
Molecular Weight:
227.23
Alternative Names:
(1S,5R)-CP-601927
- Data sheet: View or download
- MSDS: View or download
- Protocol: View or download
Product Description:
CP-601932 ((1S,5R)-CP-601927) is a high-affinity partial agonist at α3β4 nAChR (Ki=21 nM; EC50=~ 3 µM). CP-601932 has the same high-binding affinity at α4β2 nAChR (Ki=21 nM) and an order of magnitude lower affinity for α6 and α7 nAChR subtypes. CP-601932 selectively decreases ethanol but not sucrose consumption and operant self-administration following long-term exposure. CP-601932 can penetrate the CNS[1].
Storage Temperature:
-20°C, 3 years; 4°C, 2 years (Powder)