This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:
1044535-52-5
Purity:
99.9
Molecular Weight:
494.55
Alternative Names:
PF-00251802
- Data sheet: View or download
- MSDS: View or download
- Protocol: View or download
Product Description:
Dagrocorat (PF-00251802) is an orally active and selective high-affinity partial agonist of the glucocorticoid receptor. Dagrocorat is also a time-dependent reversible inhibitor of CYP3A (IC50=1.3 µM in human liver microsomes) and CYP2D6 (Ki=0.57 µM in human liver microsomes). Dagrocorat can be used for the research of rheumatoid arthritis[1].
Storage Temperature:
-20°C, 3 years; 4°C, 2 years (Powder)