This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:
633283-39-3
Purity:
98.7
Molecular Weight:
345.85
- Data sheet: View or download
- MSDS: View or download
- Protocol: View or download
Product Description:
VU10010 is a potent, highly selective and allosteric M4 mAChR potentiator with an EC50 of 400 nM. VU10010 binds to an allosteric site on M4 mAChR and increases affinity for acetylcholine and coupling to G proteins. VU10010 increases carbachol-induced depression of transmission at excitatory but not inhibitory synapses in the hippocampus[1].
Storage Temperature:
-20°C, 3 years; 4°C, 2 years (Powder)