This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:
1627929-55-8
Purity:
99.74
Molecular Formula:
C26H22N4O3
Molecular Weight:
438.48
- Data sheet: View or download
- MSDS: View or download
- Protocol: View or download
Product Description:
PLX51107 is a potent and selective BET inhibitor, with Kds of 1.6, 2.1, 1.7, and 5 nM for BD1 and 5.9, 6.2, 6.1, and 120 nM for BD2 of BRD2, BRD3, BRD4, and BRDT, respectively; PLX51107 also interacts with the bromodomains of CBP and EP300 (Kd, in the 100 nM range).
Storage Temperature:
-20°C, 3 years; 4°C, 2 years (Powder)