Talabostat (mesylate)
Catalogue number:
HY-13233A-10mg
Supplier:
Size:
10 mg
Product is available in:
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:
150080-09-4
Purity:
99.05
Molecular Weight:
310.18
Alternative Names:
Val-boroPro (mesylate); PT100 (mesylate)
- Data sheet: View or download
- MSDS: View or download
- Protocol: View or download
Product Description:
Talabostat mesylate (Val-boroPro mesylate; PT100 mesylate) is an orally active and nonselective dipeptidyl peptidase IV (DPP-IV) inhibitor (IC50 < 4 nM; Ki = 0.18 nM) and the first clinical inhibitor of fibroblast activation protein (FAP) (IC50 = 560 nM), inhibits DPP8/9 (IC50 = 4/11 nM; Ki = 1.5/0.76 nM), quiescent cell proline dipeptidase (QPP) (IC50 = 310 nM), DPP2, and some other DASH family enzymes. Antineoplastic and hematopoiesis- stimulating activities[1][2][3].
Storage Temperature:
4°C (Powder, sealed storage, away from moisture)