This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:
871362-31-1
Purity:
99.19
Molecular Weight:
391.77
Alternative Names:
RO 4956371; mGluR5 inhibitor
- Data sheet: View or download
- MSDS: View or download
- Protocol: View or download
Product Description:
CTEP (RO 4956371) is a novel, long-acting, orally bioavailable allosteric antagonist of?mGlu5?receptor with?IC50?of 2.2 nM, and shows > 1000-fold selectivity over other mGlu receptors. CTEP is a click chemistry reagent, itcontains an Alkyne group and can undergo copper-catalyzed azide-alkyne cycloaddition (CuAAc) with molecules containing Azide groups.
Storage Temperature:
4°C (Powder, sealed storage, away from moisture and light)