Aprocitentan
Catalogue number:
HY-15895-100mg
Supplier:
Size:
100 mg
Product is available in:
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:
1103522-45-7
Purity:
99.98
Molecular Weight:
546.19
Alternative Names:
ACT-132577
- Data sheet: View or download
- MSDS: View or download
- Protocol: View or download
Product Description:
Aprocitentan (ACT-132577) is the major and pharmacologically active metabolite of Macitentan. Aprocitentan is dual ETA/ETB antagonist with IC50s of 3.4 nM and 987 nM, and pA2 valus of 6.7 and 5.5, respectively[1].
Storage Temperature:
-20°C, 3 years; 4°C, 2 years (Powder)