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PD 168568 (hydrochloride)

Catalogue number:
CAY35483-5 mg
Supplier:
Size:
5 mg
Product is available in:
  • UK
  • Ireland
  • Europe
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  • Rest of World
£139.00 Estimated delivery Wed 7 Aug
Shipping is calculated in checkout
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:

1782532-06-2

Purity:

≥98%

Formulation:

A solid

Molecular Weight:

422.4

Alternative Names:

3-[2-[4-(3,4-dimethylphenyl)-1-piperazinyl]ethyl]-2,3-dihydro-1h-isoindol-1-one, dihydrochloride

Product Description:

A dopamine D4 receptor antagonist (Ki = 8.8 nM); selective for dopamine D4 over D2 receptors (Ki = 1,842 nM); reverses amphetamine-induced hyperlocomotion in rats at 3 mg/kg; inhibits the growth of glioblastoma neural stem cells at 25 and 50 µM

Storage Temperature:

-20°C

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