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MK-4827 (tosylate)

Catalogue number:
CAY20842-50 mg
Supplier:
Size:
50 mg
Product is available in:
  • UK
  • Ireland
  • Europe
  • USA
  • Rest of World
£328.00 Estimated delivery Wed 7 Aug
Shipping is calculated in checkout
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:

1038915-73-9

Purity:

≥98%

Formulation:

A crystalline solid

Molecular Weight:

492.6

Alternative Names:

2-[4-(3s)-3-piperidinylphenyl]-2h-indazole-7-carboxamide, 4-methylbenzenesulfonate, niraparib tosylate

Product Description:

An orally bioavailable inhibitor of PARP1 and PARP2 (IC50s = 3.8 and 2.1 nM, respectively); inhibits the proliferation of BRCA1 and BRCA2 mutant cancer cells in vitro (IC50s = 10-100 nM) and has efficacy alone against a xenograft of BRCA1-deficient cancer in mice

Storage Temperature:

-20°C

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