O-Desmethyl gefitinib-d8
Catalogue number:
HY-100064S-1mg
Supplier:
Size:
1 mg _$$_
Product is available in:
This product is for research use only and is not for human consumption or therapeutic use.
Purity:
99.84
Molecular Formula:
C21H14D8ClFN4O3
Molecular Weight:
440.93
- Data sheet: View or download
- MSDS: View or download
- Protocol: View or download
Product Description:
O-Desmethyl gefitinib-d8 is a deuterium labeled O-Desmethyl gefitinib. O-Desmethyl gefitinib is an active metabolite of Gefitinib in human plasma. The formation of O-desmethyl gefitinib is dependent on CYP2D6 activity. O-desmethyl gefitinib inhibits EGFR with an IC50 of 36 nM in subcellular assays[1][2].
Storage Temperature:
-20°C, 3 years; 4°C, 2 years (Powder)