NAS-181 (dimesylate)
Catalogue number:
HY-103156-5mg
Supplier:
Size:
5 mg _$$_
Product is available in:
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:
1217474-40-2
Purity:
98.44
Molecular Formula:
C21H34N2O10S2
Molecular Weight:
538.63
- Data sheet: View or download
- MSDS: View or download
- Protocol: View or download
Product Description:
NAS181 is a potent and selective antagonist of rat 5-HT1B receptor, with a Ki of 47 nM. NAS181 shows 13-fold selectivity for r5-HT1B over bovine 5-HT1B receptor (Ki=630 nM). NAS181 increases the 5-HT turnover and the synaptic concentration of 5-HT by inhibiting terminal r5-HT1B autoreceptors[1][2].
Storage Temperature:
4°C (Powder, sealed storage, away from moisture)