This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:
213027-19-1
Purity:
99.26
Molecular Weight:
216.32
Alternative Names:
GT-2331
- Data sheet: View or download
- MSDS: View or download
- Protocol: View or download
Product Description:
Cipralisant (GT-2331) is an orally active, low-toxicity, potent, selective, high affinity histamine H3 receptor full antagonist in vivo, and an agonist in vitro, with a pKi of 9.9 for histamine H3 receptor and a Ki of 0.47 nM for rat histamine H3 receptor. Cipralisant has the potential for attention-deficit hyperactivity disorder research[1][2][3][4]. Cipralisant is a click chemistry reagent, itcontains an Alkyne group and can undergo copper-catalyzed azide-alkyne cycloaddition (CuAAc) with molecules containing Azide groups.
Storage Temperature:
-20°C, 3 years; 4°C, 2 years (Powder)