(S)-(+)-Dimethindene (maleate)
Catalogue number:
HY-107647-25mg
Supplier:
Size:
25 mg _$$_
Product is available in:
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:
136152-65-3
Purity:
99.94
Molecular Weight:
408.49
- Data sheet: View or download
- MSDS: View or download
- Protocol: View or download
Product Description:
(S)-(+)-Dimethindene maleate, an enantiomer, is a potent M2-selective muscarinic receptor antagonist (pA2 = 7.86/7.74; pKi = 7.78). (S)-(+)-Dimethindene maleate shows lower affinities for the muscarinic M1 (pA2 = 6.83/6.36; pKi = 7.08), the M3 (pA2 = 6.92/6.96; pKi = 6.70) and the M4 receptors (pKi = 7.00), respectively. (S)-(+)-Dimethindene maleate also is a histamine H1 receptor antagonist (pA2 = 7.48)[1].
Storage Temperature:
4°C (Powder, sealed storage, away from moisture)