Opiranserin (hydrochloride)
Catalogue number:
HY-109067A-100mg
Supplier:
Size:
100 mg _$$_
Product is available in:
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:
1440796-75-7
Purity:
99.44
Molecular Weight:
430.97
Alternative Names:
VVZ-149 (hydrochloride)
- Data sheet: View or download
- MSDS: View or download
- Protocol: View or download
Product Description:
Opiranserin (VVZ-149) hydrochloride, a non-opioid and non-NSAID analgesic candidate, is a dual antagonist of glycine transporter type 2 (GlyT2) and serotonin receptor 2A (5HT2A), with IC50s of 0.86 and 1.3 µM, respectively. Opiranserin hydrochloride shows antagonistic activity on rP2X3 (IC50=0.87 µM). Opiranserin hydrochloride is development as an injectable agent for the treatment of postoperative pain[1][2][3].
Storage Temperature:
-20°C, 3 years; 4°C, 2 years (Powder)