This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:
1239729-06-6
Purity:
98.29
Molecular Weight:
450.36
Alternative Names:
RP5063
- Data sheet: View or download
- MSDS: View or download
- Protocol: View or download
Product Description:
Brilaroxazine (RP5603) is a potent and orally active multimodal dopamine (DA)/serotonin (5-HT) modulator. Brilaroxazine is a partial agonist of dopamine (DA) D2, D3, and D4 receptors, 5-HT1A (Ki=1.5 nM) and 5-HT2A (Ki=2.5 nM), and has antagonist activity at 5-HT2B (Ki=0.19 nM), and 5-HT7 (Ki=2.7 nM) receptors[1]. Brilaroxazine is an atypical antipsychotic agent, and has the potential to improve cognitive impairments in neuropsychiatric and neurological diseases in vivo[2].
Storage Temperature:
4°C (Powder, protect from light)