This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:
877387-37-6
Purity:
99.85
Molecular Weight:
417.55
- Data sheet: View or download
- MSDS: View or download
- Protocol: View or download
Product Description:
GSK5182 is a highly selective and orally active inverse agonist of estrogen-related receptor γ (ERRγ) with an IC50 of 79 nM. GSK5182 does not interact with other nuclear receptors, including ERRα or ERα. GSK5182 also induces reactive oxyen species (ROS) generation in hepatocellular carcinoma (HCC)[1][2][3].
Storage Temperature:
-20°C, 3 years; 4°C, 2 years (Powder)