This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:
862892-90-8
Purity:
99.11
Molecular Formula:
C10H13ClN4O2
Molecular Weight:
256.69
- Data sheet: View or download
- MSDS: View or download
- Protocol: View or download
Product Description:
GSK256073 is a potent, selective and orally active GPR109A agonist and a long-lasting and non-flushing HCA2 full agonist with a pEC50 of 7.5 (human HCA2). GSK256073 acutely improves glucose homeostasis via inhibition of lipolysis and has the potential for the study of type 2 diabetes mellitus (T2DM)and dyslipidemia[1][2]. GPR109A: G-protein coupled receptor 109A; HCA2: hydroxy-carboxylic acid receptor 2
Storage Temperature:
-20°C, 3 years; 4°C, 2 years (Powder)