UCSF924
Catalogue number:
HY-125751-50mg
Supplier:
Size:
50 mg
Product is available in:
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:
1434515-70-4
Purity:
99.56
Molecular Weight:
322.4
- Data sheet: View or download
- MSDS: View or download
- Protocol: View or download
Product Description:
UCSF924 is a potent and specific dopamine D4 receptor (DRD4) partial agonist with a EC50 of 4.2 nM. UCSF924 has a high-affinity with a Ki value of 3 nM for DRD4 and shows no measurable affinity for D2, D3 or the F261V/L328F D4 mutant. UCSF924 is a 7.4-fold bias toward arrestin over Gαi/o signaling, referenced to quinpirole[1].
Storage Temperature:
-20°C, 3 years; 4°C, 2 years (Powder)