This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:
1973403-00-7
Purity:
99.9
Molecular Formula:
C53H56F3N7O7S2
Molecular Weight:
1024.18
- Data sheet: View or download
- MSDS: View or download
- Protocol: View or download
Product Description:
ARCC-4 is a low-nanomolar Androgen Receptor (AR) degrader based on PROTAC, with a DC50 of 5 nM. ARCC-4 is an enzalutamide-based von Hippel-Lindau (VHL)-recruiting AR PROTAC and outperforms enzalutamide. ARCC-4 effectively degrades clinically relevant AR mutants associated with antiandrogen therapy[1].
Storage Temperature:
-20°C, 3 years; 4°C, 2 years (Powder)