BET bromodomain inhibitor 1
Catalogue number:
HY-131061-100mg
Supplier:
Size:
100 mg _$$_
Product is available in:
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:
2411226-02-1
Purity:
99.91
Molecular Formula:
C22H19F2N3O4S
Molecular Weight:
459.47
- Data sheet: View or download
- MSDS: View or download
- Protocol: View or download
Product Description:
BET bromodomain inhibitor 1 is an orally active, selective bromodomain and extra-terminal (BET) bromodomain inhibitor with an IC50 of 2.6 nM for BRD4. BET bromodomain inhibitor 1 binds to BRD2(2), BRD3(2), BRD4(1), BRD4(2), and BRDT(2) with high affinities (Kd values of 1.3 nM, 1.0 nM, 3.0 nM, 1.6 nM, 2.1 nM, respectively). bromodomain inhibitor 1 has anti-cancer activity[1].
Storage Temperature:
-20°C, 3 years; 4°C, 2 years (Powder)