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ERα degrader-2

Catalogue number:
HY-132194-10mg
Supplier:
Size:
10 mg _$$_
Product is available in:
  • UK
  • Ireland
  • Europe
  • USA
  • Rest of World
£870.00 Shipping is calculated in checkout
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:

2235396-63-9

Purity:

99.71

Molecular Formula:

C29H27F3N2O2

Molecular Weight:

492.53

Product Description:

ERα degrader-2 is a selective estrogen receptor degrader (SERD) with potent binding affinity with ERα (IC50=17.1 nM), good degradation efficacy (EC50=0.3 nM). ERα degrader-2 exhibits favorable pharmacokinetic properties and excellent agentgability, can be used for HER+ breast cancer research[1].

Storage Temperature:

4°C (Powder, sealed storage, away from moisture and light)

Details Cat number & supplier Size Price
ERα degrader-2 HY-132194-100mg · MedChem Express
HY-132194-100mg
MedChem Express
100 mg £5590.00
100 mg
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ERα degrader-2 HY-132194-25mg · MedChem Express
HY-132194-25mg
MedChem Express
25 mg £1839.00
25 mg
view
PD-1/PD-L1-IN-9 (hydrochloride) HY-132192A-5mg · MedChem Express
HY-132192A-5mg
MedChem Express
5 mg £435.00
5 mg
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ERα degrader-2 HY-132194-50mg · MedChem Express
HY-132194-50mg
MedChem Express
50 mg £3168.00
50 mg
view
PD-1/PD-L1-IN-9 (hydrochloride) HY-132192A-50mg · MedChem Express
HY-132192A-50mg
MedChem Express
50 mg £2113.00
50 mg
view
ERα degrader-2 HY-132194-5mg · MedChem Express
HY-132194-5mg
MedChem Express
5 mg £560.00
5 mg
view
PD-1/PD-L1-IN-9 (hydrochloride) HY-132192A-25mg · MedChem Express
HY-132192A-25mg
MedChem Express
25 mg £1367.00
25 mg
view
BTK inhibitor 18 HY-132196-100mg · MedChem Express
HY-132196-100mg
MedChem Express
100 mg £9317.00
100 mg
view
PD-1/PD-L1-IN-9 (hydrochloride) HY-132192A-10mg · MedChem Express
HY-132192A-10mg
MedChem Express
10 mg £721.00
10 mg
view
BTK inhibitor 18 HY-132196-10mg · MedChem Express
HY-132196-10mg
MedChem Express
10 mg £1839.00
10 mg
view