This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:
2651200-35-8
Purity:
99.01
Molecular Weight:
454.36
- Data sheet: View or download
- MSDS: View or download
- Protocol: View or download
Product Description:
CDK12-IN-5, a pyrazolotriazine, is a potent CDK12 inhibitor with an IC50 of 23.9 nM at high ATP (2 mM). CDK12-IN-5 has no effect on CDK2/Cyclin E (IC50=173 µM) and CDK9/Cyclin T1 (IC50=127 µM) at high ATP (2 mM) (WO2021116178A1)[1].
Storage Temperature:
-20°C, 3 years; 4°C, 2 years (Powder)