Zeteletinib
Catalogue number:
HY-139590-25mg
Supplier:
Size:
25 mg
Product is available in:
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:
2216753-97-6
Purity:
99.06
Molecular Weight:
500.47
Alternative Names:
BOS-172738; DS-5010
- Data sheet: View or download
- MSDS: View or download
- Protocol: View or download
Product Description:
Zeteletinib (BOS-172738; DS-5010) is an orally active, selective RET kinase inhibitor with nanomolar potency against RET and >300-fold selectivity against VEGFR2. Zeteletinib shows exquisite potency for the wild type RET, RETV804M/L gatekeeper mutants, and the most common oncogenic RET mutation M918T. Zeteletinib has potent antitumor activity[1][2][3].
Storage Temperature:
-20°C, 3 years; 4°C, 2 years (Powder)