CCG258747
Catalogue number:
HY-139690-10mg
Supplier:
Size:
10 mg
Product is available in:
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:
2615910-00-2
Purity:
99.17
Molecular Weight:
502.54
- Data sheet: View or download
- MSDS: View or download
- Protocol: View or download
Product Description:
CCG258747 is a selective GRK2 inhibitor (IC50=18 nM) with high selectivity over GRK1, GRK5, PKA, and ROCK1 (518, 83, >5500, and >550–fold, respectively).CCG258747 also blocks the internalization of the µ-opioid receptor. G protein-coupled receptor (GPCR) kinases (GRKs) are attractive targets for the research of heart failure[1].
Storage Temperature:
4°C (Powder, sealed storage, away from moisture and light)