I-BET151 (GSK1210151A)
Catalogue number:
BPS-27629-1
Supplier:
Size:
5 mg _$$_
Product is available in:
CAS Number:
1300031-49-5
Molecular Weight:
415.4
Product Description:
I-BET151(GSK1210151A) is a BET bromodomain inhibitor. I-BET151 displays potent binding affinity to BRD2, BRD3 and BRD4 with Kd of 0.02-0.1 µM. I-BET151 (0.5 or 5 µM) inhibits the binding of BETs (BRD2, BRD3, BRD4, and BRD9) but not the binding of 23 other bromodomain proteins. I-BET151 also blocks recruitment of BET to chromatin.
Storage Temperature:
Store at or below -20°C. Solid form is stable at least 12 months from date of receipt, when stored a
