CAS Number:
1403254-99-8
Purity:
≥99% by HPLC
Molecular Weight:
572.7
Product Description:
EPZ-6438 is a potent and bio-available inhibitor of EZH2, the catalytic subunit of polycomb repressive complex 2 (PRC2) catalyzing the methylation of lysine 27 of histone H3 (H3K27), that inhibits the activity of human PRC2-containing wild-type EZH2 (Ki = 2.5 nM).
Storage Temperature:
Store desiccated at or below -20°C. Solid form is stable at least 12 months from date of receipt, wh