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K252a

Catalogue number:
Supplier:
Size:
1 mg _$$_
Product is available in:
  • UK
  • Ireland
  • Europe
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£266.00 Shipping is calculated in checkout
CAS Number:

97161-97-2

Purity:

≥99%

Molecular Weight:

467.5

Product Description:

K252a is a general kinase inhibitor that inhibits PKA (Ki = 18 nM), PKC (Ki = 25 nM), PKG (Ki = 20 nM), CaMK (Ki = 1.8 nM), and phosphorylase kinase (IC50 = 1.7 nM). It functions by acting competitively with ATP and noncompetitively with the substrate.

Storage Temperature:

Store at or below -20°C. Solid form is stable at least 12 months from date of receipt, when stored a

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