Promethazine (hydrochloride)
Catalogue number:
CAY16478-25 g
Supplier:
Size:
25 g
Product is available in:
£69.00
Estimated delivery Wed 7 Aug
Shipping is calculated in checkout
Shipping is calculated in checkout
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:
58-33-3
Purity:
≥95%
Formulation:
A crystalline solid
Molecular Weight:
320.9
Alternative Names:
n,n,α-trimethyl-10h-phenothiazine-10-ethanamine, monohydrochloride, nsc 231688
- Data sheet: View or download
- MSDS: View or download
Product Description:
A histamine H1 receptor antagonist (Ki = 0.98 nM for the human receptor); selective for histamine H1 over H3 and H4 receptors (Kis = >100 and 77.6 µM, respectively, for the human receptors); binds mAChRs (Ki = 22 nM); inhibits histamine-induced paw edema and acetic acid-induced writhing in mice (ED50s = 5.9 and 11.8 mg/kg, respectively); decreases the number of motion-induced vomiting episodes in S. murinus at 32 mg/kg
Storage Temperature:
-20°C
