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TAK-632

Catalogue number:
CAY16285-50 mg
Supplier:
Size:
50 mg
Product is available in:
  • UK
  • Ireland
  • Europe
  • USA
  • Rest of World
£984.00 Estimated delivery Wed 7 Aug
Shipping is calculated in checkout
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:

1228591-30-7

Purity:

≥98%

Formulation:

A crystalline solid

Molecular Weight:

554.5

Alternative Names:

n-[5-[[7-cyano-2-[(cyclopropylcarbonyl)amino]-6-benzothiazolyl]oxy]-2-fluorophenyl]-3-(trifluoromethyl)-benzeneacetamide

Product Description:

A selective slow off-rate inhibitor of Raf kinases (IC50s = 8.3, 2.4, and 1.4 nM for wild type B-Raf, mutant B-RafV600E, and c-Raf, respectively); shows significant antiproliferative activity against mutated BRAF or mutated NRAS cancer cell lines and xenograft models

Storage Temperature:

-20°C

CAY16285-50 mg: TAK-632
CAY16285-50 mg: TAK-632
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