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MF63

Catalogue number:
CAY13217-1 mg
Supplier:
Size:
1 mg
Product is available in:
  • UK
  • Ireland
  • Europe
  • USA
  • Rest of World
£45.00 Estimated delivery Wed 7 Aug
Shipping is calculated in checkout
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:

892549-43-8

Purity:

≥98%

Formulation:

A crystalline solid

Molecular Weight:

378.8

Alternative Names:

2-(9-chloro-1h-phenanthro[9,10-d]imidazol-2-yl)-1,3-benzenedicarbonitrile

Product Description:

A potent, selective, and orally active inhibitor of human mPGES-1 (IC50 = 1.3 nM); potently inhibits guinea pig mPGES-1 (IC50 = 0.9 nM) but not mouse or rat mPGES-1; prevents LPS-induced pyresis, hyperalgesia, and iodoacetate-induced osteoarthritic pain

Storage Temperature:

22°C

CAY13217-1 mg: MF63
CAY13217-1 mg: MF63
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