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PF-299804

Catalogue number:
CAY9001879-50 mg
Supplier:
Size:
50 mg
Product is available in:
  • UK
  • Ireland
  • Europe
  • USA
  • Rest of World
£1377.00 Estimated delivery Wed 7 Aug
Shipping is calculated in checkout
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:

1110813-31-4

Purity:

≥98%

Formulation:

A crystalline solid

Molecular Weight:

469.9

Alternative Names:

n-[4-[(3-chloro-4-fluorophenyl)amino]-7-methoxy-6-quinazolinyl]-4-(1-piperidinyl)-(2e)-butenamide, dacomitinib, pf-299

Product Description:

An irreversible pan-ErbB receptor tyrosine kinase inhibitor (IC50s = 6, 45.7, and 73.7 nM for ErbB1, ErbB2, and ErbB4, respectively); demonstrates antitumor activity in various tumor xenograft models expressing either wild-type ErbB or mutant ErbB family members that show resistance to first generation ErbB kinase inhibitors

Storage Temperature:

-20°C

CAY9001879-50 mg: PF-299804
CAY9001879-50 mg: PF-299804
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