GSK1059615
Catalogue number:
CAY11569-50 mg
Supplier:
Size:
50 mg
Product is available in:
£592.00
Estimated delivery Wed 7 Aug
Shipping is calculated in checkout
Shipping is calculated in checkout
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:
958852-01-2
Purity:
≥98%
Formulation:
A crystalline solid
Molecular Weight:
333.4
Alternative Names:
5z-[[4-(4-pyridinyl)-6-quinolinyl]methylene]-2,4-thiazolidinedione
- Data sheet: View or download
- MSDS: View or download
Product Description:
A potent, reversible, ATP-competitive, thiazolidinedione inhibitor of PI3Kα (IC50 = 2 nM) and the common activating mutants of p100α (E542K, E545K, and H1047R) found in cancer; prevents proliferation in BT474 tumor xenografts and reduces MAPK signaling with twice daily dosing at 25 mg/kg
Storage Temperature:
-20°C
