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BRL 50481

Catalogue number:
CAY16899-25 mg
Supplier:
Size:
25 mg
Product is available in:
  • UK
  • Ireland
  • Europe
  • USA
  • Rest of World
£223.00 Estimated delivery Wed 7 Aug
Shipping is calculated in checkout
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:

433695-36-4

Purity:

≥98%

Formulation:

A crystalline solid

Molecular Weight:

244.3

Alternative Names:

n,n,2-trimethyl-5-nitro-benzenesulfonamide

Product Description:

A potent, selective inhibitor of PDE7, inhibiting human recombinant PDE7A1 with a Ki value of 180 nM; enhances the inhibitory effects of the PDE4 blocker rolipram on monocytes, lung macrophgaes, and CD8+ T-lymphocytes; promotes apoptosis in chronic lymphocytic leukemia cells overexpressing PDE7B

Storage Temperature:

-20°C

CAY16899-25 mg: BRL 50481
CAY16899-25 mg: BRL 50481
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