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CEP-33779

Catalogue number:
CAY16732-1 mg
Supplier:
Size:
1 mg
Product is available in:
  • UK
  • Ireland
  • Europe
  • USA
  • Rest of World
£142.00 Estimated delivery Wed 7 Aug
Shipping is calculated in checkout
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:

1257704-57-6

Purity:

≥95%

Formulation:

A crystalline solid

Molecular Weight:

462.6

Alternative Names:

n-[3-(4-methyl-1-piperazinyl)phenyl]-8-[4-(methylsulfonyl)phenyl]-[1,2,4]triazolo[1,5-a]pyridin-2-amine

Product Description:

A potent, orally available inhibitor of JAK2 (IC50 = 1.3 nM); reduces the production of inflammatory cytokines and blocks disease development in mouse models of lupus and arthritis; induces regression of established colorectal tumors in mice, reducing angiogenesis and proliferation of tumor cells

Storage Temperature:

-20°C

CAY16732-1 mg: CEP-33779
CAY16732-1 mg: CEP-33779
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