www.bioscience.co.uk
Sales & Support: +44 (0)1223 316 855

*

MK-0457

Catalogue number:
CAY13600-25 mg
Supplier:
Size:
25 mg
Product is available in:
  • UK
  • Ireland
  • Europe
  • USA
  • Rest of World
£112.00 Estimated delivery Wed 7 Aug
Shipping is calculated in checkout
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:

639089-54-6

Purity:

≥98%

Formulation:

A crystalline solid

Molecular Weight:

464.6

Alternative Names:

n-[4-[[4-(4-methyl-1-piperazinyl)-6-[(5-methyl-1h-pyrazol-3-yl)amino]-2-pyrimidinyl]thio]phenyl]-cyclopropanecarboxamide, tozasertib, vx-680

Product Description:

A potent pan-Aurora kinase inhibitor that favors Aurora A (Ki = 0.6 nM) over Aurora B (Ki = 18 nM) or Aurora C (Ki = 4.6 nM); inhibits proliferation of clear cell renal carcinoma (IC50 = 2/M phase

Storage Temperature:

-20°C

CAY13600-25 mg: MK-0457
CAY13600-25 mg: MK-0457
Details Cat number & supplier Size Price
ZM 306416 CAY16968-1 mg · Cayman Chemical
CAY16968-1 mg
Cayman Chemical
1 mg £58.00
1 mg
view
SB-269970 (hydrochloride) CAY17081-5 mg · Cayman Chemical
CAY17081-5 mg
Cayman Chemical
5 mg £126.00
5 mg
view
Rp-Cyclic AMPS (triethylammonium salt) CAY16985-500 ug · Cayman Chemical
CAY16985-500 ug
Cayman Chemical
500 µg £102.00
500 µg
view
GW 441756 CAY16915-1 mg · Cayman Chemical
CAY16915-1 mg
Cayman Chemical
1 mg £42.00
1 mg
view
BG45 CAY16918-5 mg · Cayman Chemical
CAY16918-5 mg
Cayman Chemical
5 mg £105.00
5 mg
view
Asiaticoside CAY11819-5 mg · Cayman Chemical
CAY11819-5 mg
Cayman Chemical
5 mg £48.00
5 mg
view
all-cis-4,7,10,13,16-Docosapentaenoic Acid CAY10008335-1 mg · Cayman Chemical
CAY10008335-1 mg
Cayman Chemical
1 mg £58.00
1 mg
view
BRD4770 CAY11787-1 mg · Cayman Chemical
CAY11787-1 mg
Cayman Chemical
1 mg £42.00
1 mg
view
BRL 50481 CAY16899-10 mg · Cayman Chemical
CAY16899-10 mg
Cayman Chemical
10 mg £102.00
10 mg
view
Biotin-azide CAY13040-1 mg · Cayman Chemical
CAY13040-1 mg
Cayman Chemical
1 mg £74.00
1 mg
view