£350.00
Estimated delivery Tue 30 Jul
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This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:
1481677-78-4
Purity:
≥95%
Formulation:
A crystalline solid
Molecular Weight:
546.7
Alternative Names:
2-(4,4-difluoropiperidin-1-yl)-n-(1-isopropylpiperidin-4-yl)-6-methoxy-7-(3-(pyrrolidin-1-yl)propoxy)quinazolin-4-amine
- Data sheet: View or download
- MSDS: View or download
Product Description:
A selective inhibitor of G9a and GLP methyltransferases that competitively inhibits binding of H3K9 substrates with a Ki = 3.7 nM; reduces H3K9 dimethylation levels in MDA-MB-231 and PANC-1 cells (IC50s = 110 and 40 nM, respectively); displays improved pharmacokinetic properties relative to UNC0638
Storage Temperature:
-20°C
