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VU0483605

Catalogue number:
CAY16941-1 mg
Supplier:
Size:
1 mg _$$_
Product is available in:
  • UK
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£64.00 Estimated delivery Tue 30 Jul
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This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:

1623101-11-0

Purity:

≥98%

Formulation:

A crystalline solid

Molecular Weight:

446.7

Alternative Names:

3-chloro-n-[3-chloro-4-(4-chloro-1,3-dihydro-1,3-dioxo-2h-isoindol-2-yl)phenyl]-2-pyridinecarboxamide

Product Description:

A selective mGluR1 PAM (EC50s = 0.39 and 0.36 µM for human and rat receptors, respectively) with no activity as a mGlu4 PAM (EC50 >10 µM); potentiates a response to glutamate in wild-type cell lines stably expressing mGlu1 and partially restores the reduction in glutamate-mediated calcium signaling in a mutant cell model of schizophrenia

Storage Temperature:

-20°C

CAY16941-1 mg: VU0483605
CAY16941-1 mg: VU0483605
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